{"id":8462,"date":"2021-12-16T13:31:28","date_gmt":"2021-12-16T18:31:28","guid":{"rendered":"https:\/\/puyapeptide.net\/product\/atosiban-cas-90779-69-4-berkualiti-tinggi-ialah-gabungan-antagonis-reseptor-contractin-dan-pressin-v1a\/"},"modified":"2021-12-16T13:31:28","modified_gmt":"2021-12-16T18:31:28","slug":"atosiban-cas-90779-69-4-berkualiti-tinggi-ialah-gabungan-antagonis-reseptor-contractin-dan-pressin-v1a","status":"publish","type":"product","link":"https:\/\/puyapeptide.net\/ms\/product\/atosiban-cas-90779-69-4-berkualiti-tinggi-ialah-gabungan-antagonis-reseptor-contractin-dan-pressin-v1a\/","title":{"rendered":"Atosiban CAS 90779-69-4 Berkualiti Tinggi ialah gabungan antagonis reseptor contractin dan pressin V1A"},"content":{"rendered":"<h2><strong>Atosiban CAS 90779-69-4 Berkualiti Tinggi ialah gabungan antagonis reseptor contractin dan pressin V1A<\/strong><\/h2>\n<p>Nama Produk: Atosiban<br \/>\nSinonim: RW-22164;RW-22164;RWJ-22164;Atosiban Impurtiy;harga atosiban;1-deamino-2d-tyr-(oet)-4-thr-8-orn- oxytocin;oxytocin,1-(3-mercaptopropanoicacid)-2-(o-ethyl-d-tyrosine)-4-l-threonine-8-l;rwj22164;ATOSIBAN ACETATE<br \/>\nCAS: 90779-69-4&lt;&amp; &gt;MF: C43H67N11O12S2<br \/>\nMW: 994.19<br \/>\nEINECS: 806-815-5<br \/>\nKategori Produk: hormon;Peptida<br \/>\nFail Mol: 90779-69-4.mol<\/p>\n<p>Atosiban ialah diperkenalkan di UK sebagai perencat suntikan kelahiran pramatang, penyebab utama morbiditi dan kematian bayi. Analog oksitosin peptida ini adalah antagonis reseptor vasopressin V1a dan reseptor oksitosin yang didapati dalam kepekatan meningkat secara mendadak dalam miometrium rahim wanita hamil dalam tempoh terdekat. Ia secara kompetitif menghalang pengecutan dalam rahim babi guinea hamil yang disebabkan oleh oxytocin dan vasopressin. Dalam percubaan terkawal plasebo berbilang pusat, dua buta, rawatan dengan atosiban menyebabkan pemanjangan kehamilan sehingga 7 hari pada wanita yang mengandung lebih daripada 28 minggu. Dalam ujian klinikal perbandingan, atosiban menunjukkan tindakan tokolitik yang setanding (pelepasan rahim) dengan ritodrine tetapi yang pertama diterima dengan lebih baik, terutamanya berkaitan dengan kesan sampingan kardiovaskular ibu. Dalam sukarelawan yang sihat, paras plasma atosiban menurun secara dwi-eksponen dengan separuh hayat awal dan tamat masing-masing 21 min dan 1.7j.<\/p>\n<p>Atosiban ialah antagonis reseptor gabungan contractin dan pressin V1A. Struktur reseptor contractin dan reseptor pressin V1A adalah serupa. Apabila reseptor hormon kontraktil disekat, hormon kontraktil masih boleh bertindak melalui reseptor V1A, jadi adalah perlu untuk menyekat dua laluan tindakan reseptor di atas apabila Buku Kimia yang sama digunakan, dan satu antagonisme tunggal reseptor boleh menghalang pengecutan rahim dengan berkesan. Ini adalah salah satu sebab utama agonis beta, penyekat saluran kalsium dan perencat sintase prostaglandin tidak berkesan menghalang pengecutan rahim.<\/p>\n<p> <strong>Atosiban CAS 90779-69-4 Sifat Kimia<\/strong><br \/>\nTakat didih 1469.0\u00b165.0 \u00b0C (Diramalkan)<br \/>\nketumpatan 1.254\u00b10.06 g\/cm3(Diramalkan)<br \/>\nsuhu storan. -20\u00b0C<br \/>\nketerlarutan H2O: \u2264100 mg\/mL<br \/>\nbentuk pepejal<br \/>\npka 12.81\u00b10.70(Diramalkan)<br \/>\nRujukan Pangkalan Data CAS 90779-69-4(Rujukan Pangkalan Data CAS)<br \/>\n&lt; &amp;&gt; <strong>Fungsi dan Penggunaan Atosiban CAS 90779-69-4<\/strong><br \/>\n1. Bersalin pramatang<br \/>\n2. Atosiban ialah agen penyekat reseptor oksitosin dalam rawatan endometriosis eksperimen dan ditunjukkan mempamerkan kecekapan terapeutik yang ketara.<\/p>\n<p>Penyelidikan Antikanser Atosiban Kesan antitumor minyak pati O. falcata telah diuji dalam tumor pepejal H22 yang dipindahkan dalam vivo . Perencatan pertumbuhan dalam tumor pepejal H22 adalah sederhana (Yang et al. 2013).<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Nama Produk: Atosiban<br \/>\nCAS: 90779-69-4<br \/>\nMF: C43H67N11O12S2<br \/>\nMW: 994.19<br \/>\nEINECS: 806-815-5<br \/>\nFail Mol: 90779-69-4.mol<\/p>\n","protected":false},"featured_media":4548,"comment_status":"open","ping_status":"closed","template":"","meta":{"om_disable_all_campaigns":false,"_monsterinsights_skip_tracking":false,"_monsterinsights_sitenote_active":false,"_monsterinsights_sitenote_note":"","_monsterinsights_sitenote_category":0,"site-sidebar-layout":"default","site-content-layout":"default","ast-site-content-layout":"default","site-content-style":"default","site-sidebar-style":"default","ast-global-header-display":"","ast-banner-title-visibility":"","ast-main-header-display":"","ast-hfb-above-header-display":"","ast-hfb-below-header-display":"","ast-hfb-mobile-header-display":"","site-post-title":"","ast-breadcrumbs-content":"","ast-featured-img":"","footer-sml-layout":"","ast-disable-related-posts":"","theme-transparent-header-meta":"default","adv-header-id-meta":"","stick-header-meta":"","header-above-stick-meta":"","header-main-stick-meta":"","header-below-stick-meta":"","astra-migrate-meta-layouts":"default","ast-page-background-enabled":"default","ast-page-background-meta":{"desktop":{"background-color":"","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-opacity":"","overlay-gradient":""},"tablet":{"background-color":"","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-opacity":"","overlay-gradient":""},"mobile":{"background-color":"","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-opacity":"","overlay-gradient":""}},"ast-content-background-meta":{"desktop":{"background-color":"var(--ast-global-color-5)","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-opacity":"","overlay-gradient":""},"tablet":{"background-color":"var(--ast-global-color-5)","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-opacity":"","overlay-gradient":""},"mobile":{"background-color":"var(--ast-global-color-5)","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-opacity":"","overlay-gradient":""}}},"product_brand":[],"product_cat":[435],"product_tag":[1225],"class_list":{"0":"post-8462","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_cat-peptida-urogenital","7":"product_tag-high-quality-atosiban-cas-90779-69-4-is-a-combined-contractin-and-pressin-v1a-receptor-antagonist-ms","8":"desktop-align-left","9":"tablet-align-left","10":"mobile-align-left","12":"first","13":"instock","14":"shipping-taxable","15":"product-type-simple"},"_links":{"self":[{"href":"https:\/\/puyapeptide.net\/ms\/wp-json\/wp\/v2\/product\/8462","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/puyapeptide.net\/ms\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/puyapeptide.net\/ms\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/puyapeptide.net\/ms\/wp-json\/wp\/v2\/comments?post=8462"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/puyapeptide.net\/ms\/wp-json\/wp\/v2\/media\/4548"}],"wp:attachment":[{"href":"https:\/\/puyapeptide.net\/ms\/wp-json\/wp\/v2\/media?parent=8462"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/puyapeptide.net\/ms\/wp-json\/wp\/v2\/product_brand?post=8462"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/puyapeptide.net\/ms\/wp-json\/wp\/v2\/product_cat?post=8462"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/puyapeptide.net\/ms\/wp-json\/wp\/v2\/product_tag?post=8462"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}