{"id":8713,"date":"2021-12-17T03:00:42","date_gmt":"2021-12-17T08:00:42","guid":{"rendered":"https:\/\/puyapeptide.net\/product\/ganirelix-asetat-cas-123246-29-7-gonadotropin-salgilatici-hormon-gnrh-antagonistleri\/"},"modified":"2021-12-17T03:00:42","modified_gmt":"2021-12-17T08:00:42","slug":"ganirelix-asetat-cas-123246-29-7-gonadotropin-salgilatici-hormon-gnrh-antagonistleri","status":"publish","type":"product","link":"https:\/\/puyapeptide.net\/tr\/product\/ganirelix-asetat-cas-123246-29-7-gonadotropin-salgilatici-hormon-gnrh-antagonistleri\/","title":{"rendered":"Ganirelix Asetat CAS 123246-29-7 Gonadotropin salg\u0131lat\u0131c\u0131 hormon (GnRH) antagonistleri"},"content":{"rendered":"<h2><strong>Ganirelix Asetat CAS 123246-29-7 Gonadotropin salg\u0131lat\u0131c\u0131 hormon (GnRH) antagonistleri<\/strong><\/h2>\n<p>\u00dcr\u00fcn Ad\u0131: Ganirelix Asetat<br \/>\nE\u015f Anlamlar\u0131: Ac-DNal-DCpa-DPal-Ser-Tyr-DHar(Et2)-Leu-Har(Et2)-Pro-DAla -NH2;Ganirelixum;ganirelix Acetate;GANIRELIX; Ganirelix Asetat USP\/EP\/BP<br \/>\nCAS: 123246-29-7<br \/>\nMF: C80H113ClN18O13<br \/>\nMW: 1570.34<br \/>\nEINECS:<br \/>\n\u00dcr\u00fcn Kategorileri: hormonlar<br \/>\nMol Dosyas\u0131: 123246-29 -7.mol<\/p>\n<p>Ganirelix asetat, endojen gonadotropin salg\u0131lat\u0131c\u0131 hormona (GnRH) (luteinize edici hormon salg\u0131lat\u0131c\u0131 hormon (LHRH) olarak da bilinir) benzer sentetik bir dekapeptit bile\u015fi\u011fidir ve rekabet\u00e7i bir \u015fekilde antagonize eden bir GnRH antagonistidir. gonadotropik GnRH resept\u00f6r\u00fc, b\u00f6ylece yolu mutasyona u\u011fratarak gonadotropin (luteinize edici hormon LH ve folik\u00fcl uyar\u0131c\u0131 hormon FSH) sekresyonunun h\u0131zl\u0131 ve geri d\u00f6n\u00fc\u015f\u00fcml\u00fc inhibisyonuna neden olur. Ganirelix asetat, hipofizden LH salg\u0131lanmas\u0131n\u0131 FSH salg\u0131lanmas\u0131ndan daha \u00f6nemli \u00f6l\u00e7\u00fcde inhibe eder, b\u00f6ylece seks hormonu \u00fcretimini azalt\u0131r.<\/p>\n<p> <strong>Ganirelix Asetat&#39;\u0131n \u0130\u015flevi ve Uygulamas\u0131 CAS 123246-29-7<\/strong><br \/>\nGanirelix asetat, ikameleri olan bir GnRH analo\u011fudur. 1, 2, 3, 6, 8 ve 10. kal\u0131nt\u0131larda. Bu bir s\u00fcperagonist de\u011fil, daha ziyade y\u00fcksek antagonist aktiviteye sahip sentetik bir dekapeptit ve pazarlanan ilk GnRH antagonistidir. Yumurtal\u0131k hiperstim\u00fclasyon do\u011furganl\u0131k tedavisi g\u00f6ren kad\u0131nlarda LH dalgalanmalar\u0131n\u0131n bask\u0131lanmas\u0131 i\u00e7in onaylanm\u0131\u015ft\u0131r; LH dalgalanmalar\u0131 normalde yumurtlamay\u0131 te\u015fvik eder. Bu ilac\u0131n amac\u0131, LH art\u0131\u015f\u0131n\u0131 bast\u0131rmak i\u00e7in gerekli ila\u00e7 g\u00fcnlerinin say\u0131s\u0131n\u0131 \u00f6nemli \u00f6l\u00e7\u00fcde azaltmak ve b\u00f6ylece yumurtal\u0131klar\u0131n yumurtal\u0131klarda kalmas\u0131n\u0131 sa\u011flamakt\u0131r. In vitro fertilizasyon (IVF) tedavi d\u00f6ng\u00fcleri, ge\u00e7mi\u015fte LH&#39;nin erken sal\u0131n\u0131m\u0131n\u0131 bast\u0131rmak i\u00e7in l\u00f6prolid asetat\u0131n uygulanmas\u0131yla ba\u015flat\u0131lm\u0131\u015ft\u0131r. Bu, yumurtlamay\u0131 engeller, b\u00f6ylece yumurtalar bir do\u011furganl\u0131k uzman\u0131 taraf\u0131ndan geri al\u0131nmak \u00fczere haz\u0131r kal\u0131r. Bu ama\u00e7la, leuprolide asetat genellikle 26 g\u00fcne kadar enjekte edilir. Klinik \u00e7al\u0131\u015fmalar, ganireliks asetat\u0131n tedaviden sadece 5 g\u00fcn sonra LH art\u0131\u015f\u0131n\u0131 durdurabildi\u011fini, LH&#39;nin bask\u0131lanmas\u0131n\u0131n FSH&#39;den daha belirgin oldu\u011funu ve daha k\u0131sa tedavi s\u00fcresinin s\u0131cak basmas\u0131 ve ba\u015f a\u011fr\u0131s\u0131 gibi ho\u015f olmayan yan etkileri en aza indirdi\u011fini g\u00f6stermi\u015ftir. .<\/p>\n<p>Genellikle klinik olarak kontroll\u00fc yumurtal\u0131k uyar\u0131m protokollerinde yard\u0131mc\u0131 \u00fcreme teknolojisi uygulanan kad\u0131nlarda erken l\u00fcteinize edici hormon zirvelerini \u00f6nlemek ve bu nedenin neden oldu\u011fu do\u011furganl\u0131k bozukluklar\u0131n\u0131n tedavisi i\u00e7in kullan\u0131l\u0131r Chemicalbook. \u0130la\u00e7 daha az yan etkiye, y\u00fcksek gebelik oranlar\u0131na ve k\u0131sa tedavi d\u00f6ng\u00fclerine sahiptir ve benzer ila\u00e7lara k\u0131yasla \u00f6nemli klinik avantajlara sahiptir.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>\u00dcr\u00fcn Ad\u0131: Ganirelix Asetat<br \/>\nCAS: 123246-29-7<br \/>\nMF: C80H113ClN18O13<br \/>\nMW: 1570.34<br \/>\n\u00dcr\u00fcn Kategorileri: hormonlar<br \/>\nMol Dosya: 123246-29-7.mol<\/p>\n","protected":false},"featured_media":2114,"comment_status":"open","ping_status":"closed","template":"","meta":{"om_disable_all_campaigns":false,"_monsterinsights_skip_tracking":false,"_monsterinsights_sitenote_active":false,"_monsterinsights_sitenote_note":"","_monsterinsights_sitenote_category":0,"site-sidebar-layout":"default","site-content-layout":"default","ast-site-content-layout":"default","site-content-style":"default","site-sidebar-style":"default","ast-global-header-display":"","ast-banner-title-visibility":"","ast-main-header-display":"","ast-hfb-above-header-display":"","ast-hfb-below-header-display":"","ast-hfb-mobile-header-display":"","site-post-title":"","ast-breadcrumbs-content":"","ast-featured-img":"","footer-sml-layout":"","ast-disable-related-posts":"","theme-transparent-header-meta":"default","adv-header-id-meta":"","stick-header-meta":"","header-above-stick-meta":"","header-main-stick-meta":"","header-below-stick-meta":"","astra-migrate-meta-layouts":"default","ast-page-background-enabled":"default","ast-page-background-meta":{"desktop":{"background-color":"","background-image":"","background-repeat":"repeat","background-position":"center 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