{"id":8800,"date":"2021-12-17T03:07:18","date_gmt":"2021-12-17T08:07:18","guid":{"rendered":"https:\/\/puyapeptide.net\/product\/puya-tedarik-degarelix-asetat-cas-214766-78-6-prostat-kanseri-tedavisinde-kullanildi\/"},"modified":"2021-12-17T03:07:18","modified_gmt":"2021-12-17T08:07:18","slug":"puya-tedarik-degarelix-asetat-cas-214766-78-6-prostat-kanseri-tedavisinde-kullanildi","status":"publish","type":"product","link":"https:\/\/puyapeptide.net\/tr\/product\/puya-tedarik-degarelix-asetat-cas-214766-78-6-prostat-kanseri-tedavisinde-kullanildi\/","title":{"rendered":"Puya Tedarik Degarelix Asetat CAS 214766-78-6 Prostat Kanseri Tedavisinde Kullan\u0131ld\u0131"},"content":{"rendered":"<h2><strong>Puya Tedarik Degarelix Asetat CAS 214766-78-6 Prostat Kanseri Tedavisinde Kullan\u0131ld\u0131<\/strong><\/h2>\n<p>\u00dcr\u00fcn Ad\u0131: DEGARELIX<br \/>\nE\u015f anlaml\u0131lar: DEGARELIX;Degarelix asetat;N-Asetil-3-(2-naftil)-D-alanil-4-kloro-D-fenilalanil-3-(3-piridil)-D -alanil-L-seril-4-[2,6-dioksoheksahidropirimidin-4(S)-ilkarboksamido]-L-fenilalanil-4-\u00fcreido-D-fenilalanil-L-leusil-N6-izopropil-L-lisil-L- prolil-D-alaninamid asetat;Degarelix asetat tuzu;D-Alaninamid, N-asetil-3-(naftalen-2-il)-D-alanil-4-kloro-D-fenilalanil-3-(piridin-3-il) -D-alanil-L-seril-4-((((4S)-2,6-dioksoheksahidropirimidin-4-il)karbonil)amino)-L-fenilalanil-4-(karbamoilamino)-D-fenilalanil-L-leusil -N6-(1-metiletil)-L-lisil-L-prolil-;Degarelix asetat(FE-200486,Degarelix);FirMagon;Degarelix, Degarelix asetat<br \/>\nCAS: 214766-78-6<br \/>\nMF: C82H103ClN18O16<br \/>\nMW: 1632.26<br \/>\nEINECS: 807-277-4<br \/>\n\u00dcr\u00fcn Kategorileri: API<br \/>\nMol Dosyas\u0131: 214766-78-6.mol<\/p>\n<p>GnRH antagonistlerinin bir prostat ve baz\u0131 meme t\u00fcrleri gibi hormonal olarak d\u00fczenlenen kanserler i\u00e7in etkili tedavi. GnRH analoglar\u0131 olarak, hipofiz bezindeki GnRH resept\u00f6rlerine rekabet\u00e7i ve geri d\u00f6n\u00fc\u015f\u00fcml\u00fc olarak ba\u011flan\u0131rlar, b\u00f6ylece l\u00fcteinize edici hormon (LH) ve folik\u00fcl uyar\u0131c\u0131 hormon (FSH) sal\u0131n\u0131m\u0131n\u0131 bloke ederler. Erkeklerde, LH&#39;nin azalmas\u0131, testislerden testosteron salg\u0131s\u0131n\u0131n ablasyonunu tetikler ve bu had\u0131m benzeri seviyeler, ilerlemi\u015f prostat kanserinin etkili y\u00f6netiminde esast\u0131r. GnRH agonistleri ile kar\u015f\u0131la\u015ft\u0131r\u0131ld\u0131\u011f\u0131nda, antagonistler, GnRH resept\u00f6r\u00fcn\u00fcn a\u015fa\u011f\u0131 reg\u00fclasyonu \u00f6ncesinde hipotalamik-hipofiz-gonadal ekseninin bir ilk uyar\u0131m\u0131 sonucunda potansiyel bir hastal\u0131k alevlenmesinden muzdarip de\u011fildir. Ayr\u0131ca, GnRH antagonistleri, dozlama sonras\u0131nda daha h\u0131zl\u0131 faydal\u0131 etkiler sa\u011flar ve gonadotropin seviyelerinin daha etkili bir \u015fekilde bask\u0131lanmas\u0131yla sonu\u00e7lan\u0131r. Bunu ak\u0131lda tutarak, degarelix asetat prostat kanseri tedavisi i\u00e7in \u00fc\u00e7\u00fcnc\u00fc nesil bir GnRH antagonisti olarak piyasaya s\u00fcr\u00fcld\u00fc ve piyasadaki di\u011fer \u00fc\u00e7\u00fcnc\u00fc nesil ajanlar olan ganireliks ve setronelix&#39;e kat\u0131l\u0131yor.<\/p>\n<p> <strong>Kimyasal \u00d6zellikleri Degarelix Asetat CAS 214766-78-6<\/strong><br \/>\nyo\u011funluk 1.325\u00b10.06 g\/cm3(\u00d6ng\u00f6r\u00fclen)<br \/>\nsaklama s\u0131cakl\u0131\u011f\u0131. Karanl\u0131k bir yerde saklay\u0131n,Atmosferde,Dondurucuda -20\u00b0C&#39;nin alt\u0131nda saklay\u0131n<br \/>\npka 10,38\u00b10,40(Tahmini)<\/p>\n<p> <strong>Degarelix Asetat CAS 214766-78-6<\/strong><br \/>\n\u0130leri hormon -ba\u011f\u0131ml\u0131 prostat karsinomu<\/p>\n<p>Desmopressin&#39; (ticari isimleri: DDAVP, DesmoMelt, Minirin, Minirin Melt, Octim, Stimate), idrar \u00fcretimini azaltan hormon olan vazopressin i\u00e7in sentetik bir ikamedir. Nazal, intraven\u00f6z veya oral veya dil alt\u0131 tableti olarak al\u0131nabilir. Doktorlar, \u015fekersiz diyabet, yatak \u0131slatma veya nokt\u00fcri tedavisi i\u00e7in en s\u0131k olarak desmopressini re\u00e7ete eder.<\/p>\n<p>Nazal, intraven\u00f6z veya tablet olarak al\u0131nabilir. Doktorlar en s\u0131k olarak \u015fekersiz diyabet veya gece idrar ka\u00e7\u0131rma tedavisi i\u00e7in Desmopressin&#39;i re\u00e7ete eder. Desmopressin&#39; (1-desamino-8-D-arginin vazopressin), dokuz amino asit i\u00e7eren bir peptit olan normal insan hormonu arginin vazopressinin modifiye edilmi\u015f bir \u015feklidir. Desmopressin&#39; asetat\u0131n t\u0131bbi kullan\u0131m\u0131 \u015funlar\u0131 i\u00e7erir: (a) yatak \u0131slatma; (b) gece idrara \u00e7\u0131kma; (c) p\u0131ht\u0131la\u015fma bozukluklar\u0131; (d) \u015fekersiz diyabet.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>\u00dcr\u00fcn Ad\u0131: DEGARELIX<br \/>\nCAS: 214766-78-6<br \/>\nMF: C82H103ClN18O16<br \/>\nMW: 1632.26<br \/>\nEINECS: 807-277-4<br \/>\n\u00dcr\u00fcn Kategorileri: API<br \/>\nMol Dosyas\u0131: 214766 -78-6.mol<\/p>\n","protected":false},"featured_media":2135,"comment_status":"open","ping_status":"closed","template":"","meta":{"om_disable_all_campaigns":false,"_monsterinsights_skip_tracking":false,"_monsterinsights_sitenote_active":false,"_monsterinsights_sitenote_note":"","_monsterinsights_sitenote_category":0,"site-sidebar-layout":"default","site-content-layout":"default","ast-site-content-layout":"default","site-content-style":"default","site-sidebar-style":"default","ast-global-header-display":"","ast-banner-title-visibility":"","ast-main-header-display":"","ast-hfb-above-header-display":"","ast-hfb-below-header-display":"","ast-hfb-mobile-header-display":"","site-post-title":"","ast-breadcrumbs-content":"","ast-featured-img":"","footer-sml-layout":"","ast-disable-related-posts":"","theme-transparent-header-meta":"default","adv-header-id-meta":"","stick-header-meta":"","header-above-stick-meta":"","header-main-stick-meta":"","header-below-stick-meta":"","astra-migrate-meta-layouts":"default","ast-page-background-enabled":"default","ast-page-background-meta":{"desktop":{"background-color":"","background-image":"","background-repeat":"repeat","background-position":"center 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