{"id":8809,"date":"2021-12-17T03:07:22","date_gmt":"2021-12-17T08:07:22","guid":{"rendered":"https:\/\/puyapeptide.net\/product\/puya-cung-cap-degarelix-axetat-cas-214766-78-6-duoc-su-dung-de-dieu-tri-ung-thu-tuyen-tien-liet\/"},"modified":"2021-12-17T03:07:22","modified_gmt":"2021-12-17T08:07:22","slug":"puya-cung-cap-degarelix-axetat-cas-214766-78-6-duoc-su-dung-de-dieu-tri-ung-thu-tuyen-tien-liet","status":"publish","type":"product","link":"https:\/\/puyapeptide.net\/vi\/product\/puya-cung-cap-degarelix-axetat-cas-214766-78-6-duoc-su-dung-de-dieu-tri-ung-thu-tuyen-tien-liet\/","title":{"rendered":"Puya cung c\u1ea5p Degarelix axetat CAS 214766-78-6 \u0111\u01b0\u1ee3c s\u1eed d\u1ee5ng \u0111\u1ec3 \u0111i\u1ec1u tr\u1ecb ung th\u01b0 tuy\u1ebfn ti\u1ec1n li\u1ec7t"},"content":{"rendered":"<h2><strong>Puya cung c\u1ea5p Degarelix axetat CAS 214766-78-6 \u0111\u01b0\u1ee3c s\u1eed d\u1ee5ng \u0111\u1ec3 \u0111i\u1ec1u tr\u1ecb ung th\u01b0 tuy\u1ebfn ti\u1ec1n li\u1ec7t<\/strong><\/h2>\n<p> T\u00ean s\u1ea3n ph\u1ea9m: DEGARELIX<br \/>\n T\u1eeb \u0111\u1ed3ng ngh\u0129a: DEGARELIX; Degarelix axetat; N-Acetyl-3- (2-naphthyl) -D-alanyl-4-chloro-D-phenylalanyl-3- (3-pyridyl) -D -alanyl-L-seryl-4- [2,6-dioxohexahydropyrimidin-4 (S) -ylcarboxamido] -L-phenylalanyl-4-ureido-D-phenylalanyl-L-leucyl-N6-isopropyl-L-lysyl-L- prolyl-D-alaninamit axetat; Mu\u1ed1i Degarelix axetat; D-Alaninamit, N-axetyl-3- (naphtalen-2-yl) -D-alanyl-4-clo-D-phenylalanyl-3- (pyridin-3-yl) -D-alanyl-L-seryl-4 &#8211; ((((4S) -2,6-dioxohexahydropyrimidin-4-yl) cacbonyl) amino) -L-phenylalanyl-4- (carbamoylamino) -D-phenylalanyl-L-leucyl -N6- (1-metylethyl) -L-lysyl-L-prolyl-; Degarelix axetat (FE-200486, Degarelix); FirMagon; Degarelix, Degarelix axetat<br \/>\n CAS: 214766-78-6<br \/>\n MF: C82H103ClN18O16<br \/>\n MW: 1632.26<br \/>\n EINECS: 807-277-4<br \/>\n Danh m\u1ee5c s\u1ea3n ph\u1ea9m: API<br \/>\n Mol File: 214766-78-6.mol <\/p>\n<p> C\u00e1c ch\u1ea5t \u0111\u1ed1i kh\u00e1ng c\u1ee7a GnRH \u0111\u00e3 \u0111\u01b0\u1ee3c ch\u1ee9ng minh l\u00e0 m\u1ed9t li\u1ec7u ph\u00e1p hi\u1ec7u qu\u1ea3 cho c\u00e1c b\u1ec7nh ung th\u01b0 \u0111\u01b0\u1ee3c \u0111i\u1ec1u ch\u1ec9nh b\u1eb1ng n\u1ed9i ti\u1ebft t\u1ed1, ch\u1eb3ng h\u1ea1n nh\u01b0 tuy\u1ebfn ti\u1ec1n li\u1ec7t v\u00e0 m\u1ed9t s\u1ed1 lo\u1ea1i v\u00fa. L\u00e0 c\u00e1c ch\u1ea5t t\u01b0\u01a1ng t\u1ef1 c\u1ee7a GnRH, ch\u00fang li\u00ean k\u1ebft c\u1ea1nh tranh v\u00e0 thu\u1eadn ngh\u1ecbch v\u1edbi c\u00e1c th\u1ee5 th\u1ec3 GnRH trong tuy\u1ebfn y\u00ean, do \u0111\u00f3 ng\u0103n ch\u1eb7n vi\u1ec7c gi\u1ea3i ph\u00f3ng hormone ho\u00e0ng th\u1ec3 h\u00f3a (LH) v\u00e0 hormone k\u00edch th\u00edch nang tr\u1ee9ng (FSH). \u1ede nam gi\u1edbi, vi\u1ec7c gi\u1ea3m LH k\u00edch ho\u1ea1t qu\u00e1 tr\u00ecnh b\u00e0i ti\u1ebft testosterone t\u1eeb tinh ho\u00e0n b\u1ecb c\u1eaft b\u1ecf, v\u00e0 m\u1ee9c \u0111\u1ed9 gi\u1ed1ng nh\u01b0 thi\u1ebfn n\u00e0y r\u1ea5t c\u1ea7n thi\u1ebft trong vi\u1ec7c ki\u1ec3m so\u00e1t hi\u1ec7u qu\u1ea3 b\u1ec7nh ung th\u01b0 tuy\u1ebfn ti\u1ec1n li\u1ec7t giai \u0111o\u1ea1n cu\u1ed1i. So v\u1edbi c\u00e1c thu\u1ed1c ch\u1ee7 v\u1eadn GnRH, thu\u1ed1c \u0111\u1ed1i kh\u00e1ng kh\u00f4ng b\u1ecb b\u00f9ng ph\u00e1t ti\u1ec1m \u1ea9n b\u1ec7nh do k\u00edch th\u00edch ban \u0111\u1ea7u c\u1ee7a tr\u1ee5c d\u01b0\u1edbi \u0111\u1ed3i-tuy\u1ebfn y\u00ean-tuy\u1ebfn sinh d\u1ee5c tr\u01b0\u1edbc khi \u0111i\u1ec1u h\u00f2a xu\u1ed1ng c\u1ee7a th\u1ee5 th\u1ec3 GnRH. H\u01a1n n\u1eefa, c\u00e1c ch\u1ea5t \u0111\u1ed1i kh\u00e1ng GnRH cung c\u1ea5p c\u00e1c t\u00e1c d\u1ee5ng c\u00f3 l\u1ee3i nhanh h\u01a1n sau khi u\u1ed1ng thu\u1ed1c v\u00e0 d\u1eabn \u0111\u1ebfn vi\u1ec7c \u1ee9c ch\u1ebf m\u1ee9c gonadotropin hi\u1ec7u qu\u1ea3 h\u01a1n. V\u1edbi suy ngh\u0129 n\u00e0y, degarelix axetat \u0111\u00e3 \u0111\u01b0\u1ee3c \u0111\u01b0a ra nh\u01b0 m\u1ed9t ch\u1ea5t \u0111\u1ed1i kh\u00e1ng GnRH th\u1ebf h\u1ec7 th\u1ee9 ba \u0111\u1ec3 \u0111i\u1ec1u tr\u1ecb ung th\u01b0 tuy\u1ebfn ti\u1ec1n li\u1ec7t v\u00e0 n\u00f3 tham gia c\u00f9ng v\u1edbi c\u00e1c ch\u1ea5t th\u1ebf h\u1ec7 th\u1ee9 ba kh\u00e1c, ganirelix v\u00e0 cetronelix, tr\u00ean th\u1ecb tr\u01b0\u1eddng. <\/p>\n<p> <strong>T\u00ednh ch\u1ea5t h\u00f3a h\u1ecdc c\u1ee7a Degarelix Acetate CAS 214766-78-6<\/strong><br \/>\n m\u1eadt \u0111\u1ed9 1.325 \u00b1 0.06 g \/ cm3 (D\u1ef1 \u0111o\u00e1n)<br \/>\n nhi\u1ec7t \u0111\u1ed9 l\u01b0u tr\u1eef. Gi\u1eef \u1edf n\u01a1i t\u1ed1i, kh\u00f4ng kh\u00ed tr\u01a1, B\u1ea3o qu\u1ea3n trong t\u1ee7 \u0111\u00f4ng, d\u01b0\u1edbi -20 \u00b0 C<br \/>\n pka 10,38 \u00b1 0,40 (D\u1ef1 \u0111o\u00e1n) <\/p>\n<p> <strong>Ch\u1ee9c n\u0103ng v\u00e0 \u1ee9ng d\u1ee5ng c\u1ee7a Degarelix Acetate CAS 214766-78-6<\/strong><br \/>\n Hormone n\u00e2ng cao &#8211; Ung th\u01b0 bi\u1ec3u m\u00f4 tuy\u1ebfn ti\u1ec1n li\u1ec7t ph\u1ee5 thu\u1ed9c <\/p>\n<p> Desmopressin &#39;(t\u00ean th\u01b0\u01a1ng m\u1ea1i: DDAVP, DesmoMelt, Minirin, Minirin Melt, Octim, Stim) l\u00e0 m\u1ed9t ch\u1ea5t thay th\u1ebf t\u1ed5ng h\u1ee3p cho vasopressin, hormone l\u00e0m gi\u1ea3m s\u1ea3n xu\u1ea5t n\u01b0\u1edbc ti\u1ec3u. N\u00f3 c\u00f3 th\u1ec3 \u0111\u01b0\u1ee3c d\u00f9ng qua \u0111\u01b0\u1eddng m\u0169i, \u0111\u01b0\u1eddng ti\u00eam t\u0129nh m\u1ea1ch, ho\u1eb7c d\u01b0\u1edbi d\u1ea1ng vi\u00ean u\u1ed1ng ho\u1eb7c ng\u1eadm d\u01b0\u1edbi l\u01b0\u1ee1i. C\u00e1c b\u00e1c s\u0129 k\u00ea \u0111\u01a1n desmopressin &#39;th\u01b0\u1eddng xuy\u00ean nh\u1ea5t \u0111\u1ec3 \u0111i\u1ec1u tr\u1ecb \u0111\u00e1i th\u00e1o nh\u1ea1t, \u0111\u00e1i d\u1ea7m ho\u1eb7c ti\u1ec3u \u0111\u00eam. <\/p>\n<p> N\u00f3 c\u00f3 th\u1ec3 \u0111\u01b0\u1ee3c d\u00f9ng qua \u0111\u01b0\u1eddng m\u0169i, ti\u00eam t\u0129nh m\u1ea1ch ho\u1eb7c d\u01b0\u1edbi d\u1ea1ng vi\u00ean n\u00e9n. C\u00e1c b\u00e1c s\u0129 k\u00ea \u0111\u01a1n Desmopressin &#39;th\u01b0\u1eddng xuy\u00ean nh\u1ea5t \u0111\u1ec3 \u0111i\u1ec1u tr\u1ecb \u0111\u00e1i th\u00e1o nh\u1ea1t ho\u1eb7c \u0111\u00e1i d\u1ea7m ban \u0111\u00eam. Desmopressin &#39;(1-desamino-8-D-arginine vasopressin) l\u00e0 m\u1ed9t d\u1ea1ng bi\u1ebfn \u0111\u1ed5i c\u1ee7a hormone arginine vasopressin b\u00ecnh th\u01b0\u1eddng c\u1ee7a con ng\u01b0\u1eddi, m\u1ed9t peptit ch\u1ee9a ch\u00edn axit amin. S\u1eed d\u1ee5ng Desmopressin &#39;acetate trong y t\u1ebf bao g\u1ed3m: (a) l\u00e0m \u01b0\u1edbt gi\u01b0\u1eddng; (b) \u0111i ti\u1ec3u \u0111\u00eam; (c) r\u1ed1i lo\u1ea1n \u0111\u00f4ng m\u00e1u; (d) \u0111\u00e1i th\u00e1o nh\u1ea1t.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>T\u00ean s\u1ea3n ph\u1ea9m: DEGARELIX<br \/>\n CAS: 214766-78-6<br \/>\n MF: C82H103ClN18O16<br \/>\n MW: 1632.26<br \/>\n EINECS: 807-277-4<br \/>\n Danh m\u1ee5c s\u1ea3n ph\u1ea9m: API<br \/>\n Mol File: 214766 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